10.下列何者藥物能最有效控制 apixaban 所造成的嚴重出血?
(A)andexanet alfa
(B)protamine
(C)vitamin K1
(D)idarucizumab
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統計: A(909), B(49), C(77), D(55), E(0) #3818645
統計: A(909), B(49), C(77), D(55), E(0) #3818645
詳解 (共 8 筆)
#7334110
抗凝血藥物解毒劑
(A)Andexanet alfa:用在Apixaban, Rivaroxaban中毒(xa找xa)
(B)Protamine:為Heparin解毒劑(Protamine帶正電,protamine帶負電,屬於化學性拮抗)
(C)Vitamin K1:用在warfarin中毒
(D)Idarucizumab:用在Dabigatran中毒(為P-gp受質)
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#7435460
抗凝血解毒劑
- Heparin (間接的IIa/Xa抑制劑) → Protamine 魚精蛋白
- Dabigatran (直接的IIa抑制劑) → Idarucizumab
- Rivaroxaban, Apixaban, Edoxaban, Betrixaban (直接的Xa抑制劑) → Andexanet alfa
- Warfarin (Vit. K epoxide reductase抑制劑) → Vit. K (Phytonadione)
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